Emapunil - CAS 226954-04-7
Catalog number:
226954-04-7
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C23H23N5O2
Molecular Weight:
401.46
COA:
Inquire
Targets:
Others
Description:
Exhibits high affinity for TSPO in rat whole brain (Ki = 0.297 nM), and high potency against human and rat glial TSPO (IC50 values are 2.73 and 3.04 nM respectively). Displays no noticeable binding to a number of other receptors, transporters or ion channels. Also displays anxiolytic and antidepressant effects in rodent models, without inducing benzodiazepine-like adverse effects.
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Purity:
>98%
Synonyms:
AC-5216; XBD-173
MSDS:
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CAS 226954-04-7 Emapunil

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