Elzasonan hydrochloride - CAS 220322-05-4
Catalog number:
220322-05-4
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C22H24Cl3N3OS
Molecular Weight:
484.86
COA:
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Targets:
5-HT Receptor
Description:
Elzasonan, also called as CP 448187, exhibits potent and selective antagonism of 5-HT1B receptors in vitro, and preclinical in vivo studies demonstrate enhanced 5-HT neurotransmission. Elzasonan is able to improve signaling to limbic regions like the hippocampus and prefrontal cortex and ultimately resulting in antidepressant effects.
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Purity:
>98%
Appearance:
Solid powder
Synonyms:
(2Z)-4-(3,4-dichlorophenyl)-2-[[2-(4-methylpiperazin-1-yl)phenyl]methylidene]thiomorpholin-3-one;hydrochloride; Elzasonan hydrochloride; Elzasonan HCl; UNII-X38F62RR8L
MSDS:
Inquire
InChIKey:
NMTRXBJYASHMND-UXTSPRGOSA-N
InChI:
1S/C22H23Cl2N3OS.ClH/c1-25-8-10-26(11-9-25)20-5-3-2-4-16(20)14-21-22(28)27(12-13-29-21)17-6-7-18(23)19(24)15-17;/h2-7,14-15H,8-13H2,1H3;1H/b21-14-;
Canonical SMILES:
CN1CCN(CC1)C2=CC=CC=C2C=C3C(=O)N(CCS3)C4=CC(=C(C=C4)Cl)Cl.Cl
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