Elacestrant - CAS 722533-56-4
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C30H38N2O2
Molecular Weight:
458.63
COA:
Inquire
Targets:
Estrogen Receptor/ERR
Description:
Elacestrant, also referred to RAD1901, is a selective and orally available estrogen receptor (ERR) degrader (IC50= 48 and 870 nM for ERα and ERβ, respectively) and selective estrogen receptor modulator (SERM).
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Brife Description:
A selective and orally available estrogen receptor (ERR) degrader
Related CAS:
1349723-93-8 (HCl)
Synonyms:
(6R)-6-[2-[ethyl-[[4-[2-(ethylamino)ethyl]phenyl]methyl]amino]-4-methoxyphenyl]-5,6,7,8-tetrahydronaphthalen-2-ol; RAD1901; RAD-1901; RAD 1901; RAD1901 HCl salt; Elacestrant dihydrochloride
Solubility:
DMSO
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Boiling Point:
609.5±55.0 ℃ at 760 Torr
Density:
1.111±0.06 g/cm3
InChIKey:
SIFNOOUKXBRGGB-AREMUKBSSA-N
InChI:
1S/C30H38N2O2/c1-4-31-17-16-22-6-8-23(9-7-22)21-32(5-2)30-20-28(34-3)14-15-29(30)26-11-10-25-19-27(33)13-12-24(25)18-26/h6-9,12-15,19-20,26,31,33H,4-5,10-11,16-18,21H2,1-3H3/t26-/m1/s1
Canonical SMILES:
CCNCCC1=CC=C(C=C1)CN(CC)C2=C(C=CC(=C2)OC)C3CCC4=C(C3)C=CC(=C4)O
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Chemical Structure

CAS 722533-56-4 Elacestrant

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