Edonentan - CAS 210891-04-6
Catalog number: 210891-04-6
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C28H32N4O5S
Molecular Weight:
536.64
COA:
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Targets:
Endothelin Receptor
Description:
Edonentan, also known as BMS-207940, is a very potent and selective ETA endothelin receptor antagonist (Ki= 10 pM) that shows 80000-fold selective for ETA vs ETB.
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Purity:
95%
Appearance:
Solid powder
Synonyms:
N-[[2-[2-[(4,5-dimethyl-1,2-oxazol-3-yl)sulfamoyl]phenyl]-5-(1,3-oxazol-2-yl)phenyl]methyl]-N,3,3-trimethylbutanamide; Edonentan; UNII-S5016F5ZH4 ;CHEMBL383581; 210891-04-6; UNII-2CCC8CH216; Edonentan[INN]; 210891-04-6 (Edonentan); 264609-13-4 (Edonentan hydrate)
MSDS:
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Quantity:
Data not available, please inquire.
InChIKey:
ORJRYNKVKJAJPY-UHFFFAOYSA-N
InChI:
InChI=1S/C28H32N4O5S/c1-18-19(2)37-30-26(18)31-38(34,35)24-10-8-7-9-23(24)22-12-11-20(27-29-13-14-36-27)15-21(22)17-32(6)25(33)16-28(3,4)5/h7-15H,16-17H2,1-6H3,(H,30,31)
Canonical SMILES:
CC1=C(ON=C1NS(=O)(=O)C2=CC=CC=C2C3=C(C=C(C=C3)C4=NC=CO4)CN(C)C(=O)CC(C)(C)C)C
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CAS 210891-04-6 Edonentan

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