EDO-S101 - CAS 1236199-60-2
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C19H28Cl2N4O2
Molecular Weight:
415.36
COA:
Inquire
Targets:
HDAC
Description:
EDO-S101 is a pan HDAC inhibitor (IC50= 9, 9 and 25 nM for HDAC1, HDAC2 and HDAC3, respectively). EDO-S101 is a first-in-class fusion molecule that combines DNA damaging effect of bendamustine with the pan-HDACi vorinostat.
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Brife Description:
A pan HDAC inhibitor
Related CAS:
1793059-58-1 (HCl)
Synonyms:
7-[5-[bis(2-chloroethyl)amino]-1-methylbenzimidazol-2-yl]-N-hydroxyheptanamide; EDO-S101; EDO-S 101; EDO-S-101; EDO-S101 HCl; EDO-S101 hydrochloride; Tinostamustine hydrochloride
Solubility:
DMSO: ≥ 30 mg/mL
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Density:
1.27±0.1 g/cm3
InChIKey:
GISXTRIGVCKQBX-UHFFFAOYSA-N
InChI:
1S/C19H28Cl2N4O2/c1-24-17-9-8-15(25(12-10-20)13-11-21)14-16(17)22-18(24)6-4-2-3-5-7-19(26)23-27/h8-9,14,27H,2-7,10-13H2,1H3,(H,23,26)
Canonical SMILES:
CN1C2=C(C=C(C=C2)N(CCCl)CCCl)N=C1CCCCCCC(=O)NO
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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CAS 1236199-60-2 EDO-S101

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