|Targets||FGFR | VEGFR|
|Description||E 3810 dihydrochloride is a dual VEGFR/FGFR tyrosine kinase inhibitor. It suppresses the tumor angiogenesis and tumor cell proliferation via inhibiting VEGFR1, -2, and -3 and FGFR-1 and -2 kinases in the nanomolar range.|
|Brife Description||dual VEGFR/FGFR tyrosine kinase inhibitor|
|Related CAS||1058137-23-7 (free base)|
|Synonyms||E 3810 dihydrochloride; E3810 dihydrochloride; E-3810 dihydrochloride; Lucitanib dihydrochloride; 6-[7-[(1-aminocyclopropyl)methoxy]-6-methoxyquinolin-4-yl]oxy-N-methylnaphthalene-1-carboxamide dihydrochloride|
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SSR128129E free acid
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BIBF 1120 esylate
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