Drinabant - CAS 358970-97-5
Catalog number:
358970-97-5
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C23H20Cl2F2N2O2S
Molecular Weight:
497.38
COA:
Inquire
Targets:
Cannabinoid Receptor
Description:
Drinabant is a highly potent, selective antagonist for the CB1 receptor with Ki values of 0.16-0.44 nM.
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Purity:
≥98%
Appearance:
White Solid
Synonyms:
AVE-1625; N-[1-[bis(4-chlorophenyl)methyl]azetidin-3-yl]-N-(3,5-difluorophenyl)methanesulfonamide;
Solubility:
Soluble in DMSO
Storage:
Store at -20 °C
MSDS:
Inquire
Application:
Cannabinoid receptor CB1 antagonists
Quality Standard:
Enterprise standard
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly.
Quantity:
Milligrams-Grams
Density:
1.458
InChIKey:
IQQBRKLVEALROM-UHFFFAOYSA-N
InChI:
1S/C23H20Cl2F2N2O2S/c1-32(30,31)29(21-11-19(26)10-20(27)12-21)22-13-28(14-22)23(15-2-6-17(24)7-3-15)16-4-8-18(25)9-5-16/h2-12,22-23H,13-14H2,1H3
Canonical SMILES:
CS(=O)(=O)N(C1CN(C1)C(C2=CC=C(C=C2)Cl)C3=CC=C(C=C3)Cl)C4=CC(=CC(=C4)F)F
Current Developer:
Sanofi-aventis
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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CAS 358970-97-5 Drinabant

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