DMPQ dihydrochloride - CAS 1123491-15-5
Category: Inhibitor
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Molecular Formula:
C16H14N2O2.2HCl
Molecular Weight:
339.22
COA:
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Targets:
PDGFR
Description:
DMPQ dihydrochloride is a potent and selective inhibitor of human vascular β-type platelet derived growth factor receptor tyrosine kinase (PDGFRβ) (IC50 = 80 nM). It displays > 100-fold selectivity over EGFR tyrosine kinase, erbB2, p56, protein kinase A and protein kinase C.
Brife Description:
PDGFRβ inhibitor
Purity:
≥99% by HPLC
Synonyms:
5,7-Dimethoxy-3-(4-pyridinyl)quinoline dihydrochloride
MSDS:
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InChIKey:
YBBAOKYVJCNJIV-UHFFFAOYSA-N
InChI:
InChI=1S/C16H14N2O2.2ClH/c1-19-13-8-15-14(16(9-13)20-2)7-12(10-18-15)11-3-5-17-6-4-11;;/h3-10H,1-2H3;2*1H
Canonical SMILES:
COC1=CC2=NC=C(C=C2C(=C1)OC)C3=CC=NC=C3.Cl.Cl
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CAS 1123491-15-5 DMPQ dihydrochloride

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