DKM 2-93 - CAS 65836-72-8
Not Intended for Therapeutic Use. For research use only.
Category:
Inhibitor
Product Name:
DKM 2-93
Synonyms:
2-chloro-N-[(3,4-dimethoxyphenyl)methyl]acetamide
CAS Number:
65836-72-8
Description:
DKM 2-93 covalently modify the catalytic cysteine of the ubiquitin-like modifier activating enzyme 5 (UBA5), thereby inhibiting its activity as a protein that activates the ubiquitin-like protein UFM1 to UFMylate proteins (IC50= 430 μM).
Molecular Weight:
243.69
Molecular Formula:
C11H14ClNO3
COA:
Inquire
MSDS:
Inquire
Canonical SMILES:
COC1=C(C=C(C=C1)CNC(=O)CCl)OC
InChI:
1S/C11H14ClNO3/c1-15-9-4-3-8(5-10(9)16-2)7-13-11(14)6-12/h3-5H,6-7H2,1-2H3,(H,13,14)
InChIKey:
CETPWRGZGWGPSV-UHFFFAOYSA-N
Targets:
E1/E2/E3 Enzyme
Chemical Structure
CAS 65836-72-8 DKM 2-93

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