|Description||Diazoxide is a potassium channel activator that causes local relaxation in smooth muscle by increasing membrane permeability to potassium ions. The cellular release of potassium switches off voltage-gated calcium ion channels which inhibits the generation of an action potential.|
|Solubility||in methanol; slightly in dilute aqueous base; insoluble in water.|
|Storage||Store at room temperature.|
|Melting Point||330-331 °C.|
Saxitoxin is the potent neurotoxin and the best-known paralytic shellfish toxin (PST). Ingestion of saxitoxin results in numbness of the oral mucosa as quickly ...
Duocarmycin is a cytotoxic agent, used as the cytotoxic component in antibody-drug conjugates.
Ruthenium red is a polycationic dye that inhibits sarcoplasmic reticulum Ca2+ release, blocks Ca2+ uptake and release from mitochondria, and prevents Ca2+ relea...
Potent ganglioblocker, a neuronal nicotinic AChR antagonist. .
A substance which inhibits cholinesterases reversibly. Alkaloid , from plants of the Zygophyllaceae family
Muscarinic toxin 2 (MT2) is one member of a family of small peptides of 65 amino acid residues of around 7076 daltons in molecular weight derived from the venom...
Nitrarine 2HCl is a hypotensive, spasmolytic, coronary dilator, sedative in experimental arrhythmias.
β-Pompilidotoxin slows the inactivation of neuronal Navs. β-Pompilidotoxin was isolated from the venoms of two wasps, Anoplius amariensis and Batozonellus macul...
Diamine oxidase activator. Na+ channels blocker.
Quinoline alkaloid, extracted from Haplophyllum bucharicum (Rutacae)
Gramine is a naturally occurring indole alkaloid present in several plant species. Gramine may play a defensive role in these plants, since it is toxic to many ...
Dihydropyridine calcium channel blocker. Antianginal; antihypertensive.
Margatoxin (MgTx) is a component of the venom of Scorpio Centruroides margaritatus. Margatoxin preferentially inhibits voltage-dependent potassium channels Kv1....
Batrachotoxin (BTX) is an extremely potent cardiotoxic and neurotoxic steroidal alkaloid found in certain species of frogs, melyrid beetles, and birds.Batrachot...
Iron carrier Synthetic
An inhibitor of serine proteinases of broad spectrum.
Seco-Duocarmycin SA is a cytotoxic agent, used as the cytotoxic component in antibody-drug conjugates.
Potent blocker of voltage-sensitive K+ channels (IC50 values are 0.1, 1.1 and 25 nM for KV1.3, KV1.1 and KV1.2 channels) respectively). Also inhibits Ca2+-activ...
Nudicauline is extracted from plants of the Ranunculaceae family, a Alpha-Bungarotoxin neuronal nicotinic receptor.
Triterpene glycoside Extracted from Dipsacus azureas