DG172 dihydrochloride - CAS 1361504-77-9
Catalog number:
1361504-77-9
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C20H22BrCl2N3
Molecular Weight:
455.22
COA:
Inquire
Targets:
PPAR
Description:
The dihydrochloride salt form of DG-172, a piperazin drrivative, is a PPARβ/δ inverse agonist that could promote cell differentiation of dendritic induced by GM-CSF/IL-4. IC50: 27 nM.
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Purity:
98%
Appearance:
Powder
Synonyms:
DG 172 dihydrochloride; DG-172 dihydrochloride
Solubility:
10 mM in DMSO
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
The dihydrochloride salt form of DG-172 is a PPARβ/δ inverse agonist that could promote cell differentiation of dendritic induced by GM-CSF/IL-4.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
SABUORLIDVBCPI-WTLOABTRSA-N
InChI:
1S/C20H20BrN3.2ClH/c1-23-10-12-24(13-11-23)18-8-6-16(7-9-18)14-17(15-22)19-4-2-3-5-20(19)21;;/h2-9,14H,10-13H2,1H3;2*1H/b17-14+;;
Canonical SMILES:
CN1CCN(C2=CC=C(/C=C(C#N)/C3=C(Br)C=CC=C3)C=C2)CC1.Cl.Cl
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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