|Description||Dendrotoxin-I is a highly selective blocker of voltage-gated K+
channels (KV1.1 and KV1.2), as well as heteromultimeric channels containing these, with other KV1 isoforms. The inhibition effect is higher in Xenopus oocytes compared to mammalian cells.
|Solubility||Soluble in water.|
|Storage||Up to four weeks at 4°C or three months at -20°C.|
The lanthanide element from Glutaned replaces calcium in its complex with prothrombine,<br/>thus preventing the formation of thrombine and interrupting the bloo...
Dendrotoxin-I is a highly selective blocker of voltage-gated K+<br/>channels (KV1.1 and KV1.2), as well as heteromultimeric channels containing these, with othe...
Seco-Duocarmycin SA is a cytotoxic agent, used as the cytotoxic component in antibody-drug conjugates.
Synthetic, an inhibitor of high-affinity choline uptake (HAChU) in synaptosomes.
An activator of voltage-sensitive Na+ channels, a suite of cyclic polyether compounds produced naturally by a species of dinoflagellate known as Karenia brevis....
Argiotoxin blocks the glutamate responses and sensorimotor transmission in motoneurones of isolated frog spinal cord.
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Deltaline has a lycoctonine carbon-atom skeleton with four six-membered rings and three five-membered rings among; three of the six-membered rings adopt chair c...
A muscarinic receptors antagonist.
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A neuronal nicotinic AChR antagonist, blocking superior cervical sympathetic ganglion
A hypolipidemic, antiatherosclerotic, anti-inflammatory agent, with angioprotective and hepatoprotective activity; antiulcerous. Sesquiterpene lactone , from pl...
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a non specific stimulant of immunogenesis; also used for erytrocytes hemolysis and automatic leucocyte numbering. Triterpene saponine, mixture of 4 glycosides f...
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20-Hydroxyecdysone (ecdysterone or 20E) is a naturally occurring ecdysteroid hormone which controls the ecdysis (moulting) and metamorphosis of arthropods. It i...
Noscapine is often used as an antitussive medication.
Syntheticquinazolone alkaloid, inhibiting cholinesterase activity in vitro.
Artemisinin is a natural product originally isolated from plants of the genus Artemisia. It effectively kills malarial parasites of the genus Plasmodium. It is ...