|Description||DC-05 is a potent and selective non-nucleoside DNMT1 (DNA methyltransferase 1) inhibitor with IC50 of 10.3 uM. It has significant selectivity toward other AdoMet-dependent protein methyltransferases. It significantly inhibits cancer cell proliferation. It inhibitis DNMT1 by binding to DNMT1 instead of incorporating into DNA.|
|Appearance||White to off-white Solid|
|Solubility||10 mM in DMSO|
|Application||DC-05 inhibits cancer cell proliferation.|
|Quality Standard||In-house standard|
|Shelf Life||2 month in rt, long time|
|Boiling Point||667.5±55.0 °C | Condition: Press: 760 Torr|
|Density||1.23±0.1 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr|
Glucose-conjugated MGMT inhibitor
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