DBPR108 - CAS 1186426-66-3
Catalog number: 1186426-66-3
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C16H25FN4O2
Molecular Weight:
324.39
COA:
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Targets:
DPP4
Description:
DBPR108 is an IC50=15 nM DPP IV inhibitor displays a more than 3000-fold selectivity over DPP8 DPP9, FAP and DPP-II. TThe in vivo effects of DBPR108, including inhibition of plasma DPP-IV activity and suppression of blood glucose elevation, were also demonstrated. DBPR108 is a potent, selective, long-acting and safe DPP-IV inhibitor as a potential treatment of type 2 diabetes mellitus.
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Purity:
>98%
Synonyms:
DBPR-108
MSDS:
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CAS 1186426-66-3 DBPR108

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