Danirixin - CAS 954126-98-8
Catalog number:
954126-98-8
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C19H21ClFN3O4S
Molecular Weight:
441.9
COA:
Inquire
Targets:
CXCR
Description:
A small molecule, non-peptide CXCR2 antagonist; High affinity (IC50 for CXCL8 binding = 12.5 nM), selective, and reversible
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Brife Description:
A small molecule, non-peptide CXCR2 antagonist; High affinity (IC50 for CXCL8 binding = 12.5 nM), selective, and reversible
Appearance:
White to Off-White Solid
Synonyms:
GSK1325756; N-(4-chloro-2-hydroxy-3-(3-piperidinylsulfonyl)phenyl)-N'-(3-fluoro-2-methylphenyl)urea
Solubility:
DMSO: > 8 mg/mL
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
MSDS:
Inquire
Quality Standard:
In-house
Quantity:
Grams-Kilos
InChIKey:
NGYNBSHYFOFVLS-LBPRGKRZSA-N
InChI:
1S/C19H21ClFN3O4S/c1-11-14(21)5-2-6-15(11)23-19(26)24-16-8-7-13(20)18(17(16)25)29(27,28)12-4-3-9-22-10-12/h2,5-8,12,22,25H,3-4,9-10H2,1H3,(H2,23,24,26)/t12-/m0/s1
Canonical SMILES:
CC1=C(C=CC=C1F)NC(=O)NC2=C(C(=C(C=C2)Cl)S(=O)(=O)C3CCCNC3)O
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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