CYR-101 - CAS 359625-79-9
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C22H23FN2O2
Molecular Weight:
366.43
COA:
Inquire
Targets:
5-HT Receptor | Sigma Receptor
Description:
MIN-101, a novel cyclic amide derivative, is a 5-HT2A and sigma 2 receptor antagonist (Ki= 7.53 nM for 5-HT2A and 8.19 nM for sigma-2, respectively).
Brife Description:
A 5-HT2A and sigma 2 receptor antagonist (Ki= 7.53 nM for 5-HT2A and 8.19 nM for sigma-2, respectively)
Synonyms:
2-((1-(2-(4-fluorophenyl)-2-oxoethyl)piperidin-4-yl)methyl)isoindolin-1-one; CYR-101; UNII-4P31I0M3BF; MT-210; MIN101; CYR101; MT210; MIN 101; CYR 101; MT 210
Solubility:
10 mM in DMSO
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Boiling Point:
551.7±50.0 ℃ at 760 Torr
Density:
1.227±0.06 g/cm3
InChIKey:
RNRYULFRLCBRQS-UHFFFAOYSA-N
InChI:
1S/C22H23FN2O2/c23-19-7-5-17(6-8-19)21(26)15-24-11-9-16(10-12-24)13-25-14-18-3-1-2-4-20(18)22(25)27/h1-8,16H,9-15H2
Canonical SMILES:
c1ccc2c(c1)CN(C2=O)CC3CCN(CC3)CC(=O)c4ccc(cc4)F
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Chemical Structure

CAS 359625-79-9 CYR-101

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