CXCR2-IN-1 - CAS 1873376-49-8
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C19H20Cl2FN3O4S
Molecular Weight:
476.35
COA:
Inquire
Targets:
CXCR
Description:
CXCR2-IN-1 is a CXCR2 antagonists (pIC50= 9.3) with favorable central nervous system penetration property (Br/Bl>0.45).
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Brife Description:
A CXCR2 antagonists (pIC50= 9.3)
Synonyms:
1-(2-chloro-3-fluorophenyl)-3-[4-chloro-2-hydroxy-3-(1-methylpiperidin-4-yl)sulfonylphenyl]urea
Solubility:
DMSO: ≥5.4 mg/mL (Need ultrasonic and warming)
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Boiling Point:
538.1±50.0 ℃ at 760 Torr
Density:
1.528±0.06 g/cm3
InChIKey:
BJYOBCUGMDKPBM-UHFFFAOYSA-N
InChI:
1S/C19H20Cl2FN3O4S/c1-25-9-7-11(8-10-25)30(28,29)18-12(20)5-6-15(17(18)26)24-19(27)23-14-4-2-3-13(22)16(14)21/h2-6,11,26H,7-10H2,1H3,(H2,23,24,27)
Canonical SMILES:
CN1CCC(CC1)S(=O)(=O)C2=C(C=CC(=C2O)NC(=O)NC3=C(C(=CC=C3)F)Cl)Cl
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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