CP-472555 - CAS 305821-96-9
Catalog number:
305821-96-9
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C31H32N2O2
Molecular Weight:
464.24
COA:
Inquire
Targets:
Others
Description:
CP-472555 is an effective Glucocorticoid receptor agonist and probably has steroid-like anti-inflammatory properties with anti-GR and anti-obesity activity in animal models.
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Purity:
≥95%
Appearance:
Solid powder
Synonyms:
2-Phenanthrenecarboxamide, 4b,5,6,7,8,8a,9,10-octahydro-7-hydroxy-4b-(phenylmethyl)-7-(1-propyn-1-yl)-N-(3-pyridinylmethyl)-, (4bS,7R,8aR)-;
Solubility:
Soluble in DMSO
Storage:
Store at -20 °C
MSDS:
Inquire
Application:
Glucocorticoid receptor antagonists
Quality Standard:
Enterprise standard
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly.
Quantity:
Milligrams-Grams
InChIKey:
SEOPOTXFVGEDGX-UPHHSBJESA-N
InChI:
1S/C31H32N2O2/c1-2-14-30(35)15-16-31(19-23-7-4-3-5-8-23)27(20-30)12-10-25-18-26(11-13-28(25)31)29(34)33-22-24-9-6-17-32-21-24/h3-9,11,13,17-18,21,27,35H,10,12,15-16,19-20,22H2,1H3,(H,33,34)/t27-,30-,31+/m1/s1
Canonical SMILES:
CC#C[C@]1(CC[C@]2(c3ccc(cc3CC[C@@H]2C1)C(=O)NCc4cccnc4)Cc5ccccc5)O
Current Developer:
Pfizer
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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