| Molecular Formula: | |
|---|---|
| Molecular Formula | C25H21FN2O |
| Molecular Weight: | |
| Molecular Weight | 384.45 |
| COA: | |
| COA | Inquire |
| Targets: | |
| Targets | Phosphodiesterase (PDE) |
| Description: | |
| Description | CP 461, belonging to a class of novel proapoptotic drugs with antineoplastic effect, specifically inhibit cyclic GMP phosphodiesterases but not cyclooxygenase-1 or -2. |
| Purity: | |
|---|---|
| Purity | >98% |
| Appearance: | |
| Appearance | Solid powder |
| Synonyms: | |
| Synonyms | CP-461 free base; CP 461 free base; CP461 free base; N-benzyl-2-[(3Z)-6-fluoro-2-methyl-3-(pyridin-4-ylmethylidene)inden-1-yl]acetamide; UNII-824ZMS3BGL; OSI-461 free base |
| MSDS: | |
| MSDS | Inquire |
| InChIKey: | |
|---|---|
| InChIKey | NVCAMOJXQVJSOM-XKZIYDEJSA-N |
| InChI: | |
| InChI | 1S/C25H21FN2O/c1-17-22(13-18-9-11-27-12-10-18)21-8-7-20(26)14-24(21)23(17)15-25(29)28-16-19-5-3-2-4-6-19/h2-14H,15-16H2,1H3,(H,28,29)/b22-13- |
| Canonical SMILES: | |
| Canonical SMILES | CC1=C(C2=C(C1=CC3=CC=NC=C3)C=CC(=C2)F)CC(=O)NCC4=CC=CC=C4 |
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