CP-409092 - CAS 194098-25-4
Catalog number:
194098-25-4
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C17H19N3O2
Molecular Weight:
297.35
COA:
Inquire
Targets:
GABA Receptor
Description:
CP-409092 is a GABA(A) partial agonist developed for the treatment of General Anxiety Disorder (GAD) and presents an interesting phenomenon of human pharmacokinetic predictions. In vitro, CP-409092 was abroadly metabolized in rat and human systems predominantly to acid metabolite formed by oxidative deamination of the N-methyl group of CP-409092 mediated by MAO-A (as deduced from inhibition experiments).
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Purity:
>98%
Appearance:
Solid powder
Synonyms:
N-[4-(methylaminomethyl)phenyl]-4-oxo-1,5,6,7-tetrahydroindole-3-carboxamide; 4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carboxylic acid (4-methylaminomethylphenyl)amide; CP 409,092; CP 409092; CP-409,092; CP-409092; CP409,092; CP409092
MSDS:
Inquire
InChIKey:
XFJIYNUISLDNLP-UHFFFAOYSA-N
InChI:
1S/C17H19N3O2/c1-18-9-11-5-7-12(8-6-11)20-17(22)13-10-19-14-3-2-4-15(21)16(13)14/h5-8,10,18-19H,2-4,9H2,1H3,(H,20,22)
Canonical SMILES:
CNCC1=CC=C(C=C1)NC(=O)C2=CNC3=C2C(=O)CCC3
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