|Description||CP-331684 is a β3-adrenergic receptor agonist used as antidiabetic drug.|
GMC 2-83 is an atypical antipsychotic without muscarinic activity.
Methyldopa (Aldomet) is a DOPA decarboxylase competitive inhibitor with an ED50 of 21.8 mg/kg.
Nebivolol selectively inhibits β1-adrenoceptor with IC50 of 0.8 nM.
Naftopidil is a selective α1-adrenergic receptor antagonist or alpha blocker with a Ki of 58.3 nM.
Salbutamol is a short-acting agonist that specifically targets β2-adrenergic receptor to alleviate bronchospasm in conditions such as asthma and chronic obstruc...
Rec 15/2615 dihydrochloride
Rec 15/2615 dihydrochloride is a selective α1B-adrenoceptor antagonist (Ki= 0.3, 1.9 and 2.6 nM at human α1B, α1A and α1D receptors respectively) potentially fo...
O-desmethyl Mebeverine alcohol hydrochlo
O-desmethyl Mebeverine alcohol hydrochloride, a metabolite of Mebeverine, is a potent inhibitor of α1 repector, causing relaxation of the gastrointestinal tract...
Alprenolol is a non-selective Beta-Adrenergic receptor and 5-HT1A receptor antagonist for the treatment of angina pectoris.
Clenhexerol is a β-adrenergic agonist.
Yohimbine, an indolalkylamine alkaloid, blocks presynaptic alpha-2 adrenergic receptors. IC50= 0.6 μM Ki: 1.05 nM, alphaα2Areceptor
Mirabegron (formerly YM-178, trade name Myrbetriq) is a drug for the treatment of overactive bladder. It was developed by Astellas Pharma and was approved in th...
This active molecular is a β-adrenergic receptor antagonist. Levonebivolol is an enantiomer of Nebivolol which is a β1 receptor blocker with nitric oxide-potent...
Hydrocortisone-17-butyrate, a glucocorticoid compound, could be used as antiinflammatory and immunosuppresive agent.
Propranolol hydrochloride, with antihypertensive, antianginal and antiarrhythmic (class II) properties, is a non-cardioselective adrenergic-beta antagonist and ...
The hydrochloride of Nifenalol. Nifenalol is a beta-adrenoceptor antagonist used for the treatment of cardiovascular and cerebrovascular diseases such as hypert...
Landiolol is an ultra-short-acting Beta 1 adrenergic receptor antagonist using for managing supraventricular tachyarrhythmias in sepsis. It is also used as an a...
Metoprolol is a a selective β1 receptor blocker for the treatment of a variety of cardiovascular disorder.
Tulobuterol hydrochloride is a salt form of Tulobuterol, which is a long-acting beta2-adrenergic receptor agonist.
DL-Adrenaline is a hormone and a neurotransmitter secreted by the medulla of the adrenal glands.
Silodosin shows high selectivity for the alpha(1A)-AR subtype.