|Description||Conivaptan HCl is a non-peptide inhibitor of antidiuretic hormone (vasopressin receptor antagonist).|
Vasopressin antagonist 1867
Vasopressin antagonist 1867 is a selective vasopressin 1B (V1b) receptor antagonist (IC50 value 3 nM for hV1b inhibition, exhibiting >1000-fold selectivity over...
TASP 0390325 is a potent and selective vasopressin V1B receptor antagonist (IC50 = 2.22 nM for rat pituitary receptor) with no significant affinity for 85 other...
d[Cha4]-AVP is a selective and potent human vasopressin V1B receptor agonist with Ki value of 1.2 nM. It stimulates corticosterone and ACTH secretion. It shows ...
SSR 149415 is a potent and orally available vasopressin V1B antagonist (Ki = 3.7 and 1.3 nM for native and recombinant rat V1b receptors, respectively), display...
OPC-21268 is a vasopressin V1 receptor antagonist with IC50 value of 0.4 μM.
Conivaptan HCl is a non-peptide inhibitor of antidiuretic hormone (vasopressin receptor antagonist).
Fedovapagon is a potent, nonpeptidic vasopressin V2 receptor agonists (EC50 of 24 nM), demonstrated positive anti-diuretic effect in nocturia
RO-5028442 is a potent and brain-penetrant hV1a antagonist. RO-5028442 is undergoing clinical trials for autistic disorder therapy.
VPA-985, an azepine compound, has been found to be a Vasopressin receptor antagonist that could be used in some cardiovascular disease therapy like hyponatraemi...
d[leu4,Lys8]-VP is a selective vasopressin V1B receptor agonist (Ki = 0.16, 64, 100 and 3800 nM for V1B, oxytocin, V2 and V1A receptors, respectively). It exhib...
Desmopressin, a synthetic analog of the endogenous antidiuretic hormone arginine vasopressin with low vasopressor activity, is a dual antagonist of V1B and V2 r...
Tolvaptan is an orally effective nonpeptide arginine vasopressin V2 receptor antagonist with IC50 of 3 nM, used to treat hyponatremia.
Felypressin is a Vasopressin 1 agonist and has effects at all Arginine vasopressin receptor 1As. It is a non-catecholamine vasoconstrictor that is chemically re...
Conivaptan, also called as YM 087 or Vaprisol, is the first is a non-peptide inhibitor of antidiuretic hormone (vasopressin receptor antagonist) approved by Un...
Desmopressin acetate, a syntheticpeptide containing nine amino acids, is analogue of the antidiuretic hormone arginine vasopressin. Improves hemostatsis by incr...
TC OT 39
TC OT 39 is a potent non-peptide oxytocin receptor partial agonist (EC50 = 33 nM and 850 nM for the oxytocin receptor and V2 vasopressin receptor, respectively)...
OPC 31260 hydrochloride
OPC 31260 is a Vasopressin receptor antagonist marketed by Otsuka. It is a benzazepine derivative that antagonizes the binding of arginine vasopressin (AVP) to ...
Ribuvaptan is a vasopressin receptor antagonist originated by Bayer HealthCare Pharmaceuticals. Now, Ribuvaptan is still in phase I development for the treatmen...
This molecular is a polypeptide which is a Antidiuretic hormone that has been found in most mammalian species and it acts as a neurotransmitter at synapses in t...