Cobimetinib hemifumarate - CAS 1369665-02-0
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C21H21F3IN3O2.1/2C4H4O4
Molecular Weight:
589.35
COA:
Inquire
Targets:
MEK
Description:
Cobimetinib, also known as GDC-0973 and XL-518, is a novel selective MEK inhibitor, and the IC50value against MEK1 is 4.2 nM, with potential antineoplastic activity.
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Related CAS:
934660-93-2 (free base)
Synonyms:
Methanone, [3,​4-​difluoro-​2-​[(2-​fluoro-​4-​iodophenyl)​amino]​phenyl]​[3-​hydroxy-​3-​(2S)​-​2-​piperidinyl-​1-​azetidinyl]​-​, (2E)​-​2-​butenedioate (2:1)
Solubility:
DMSO
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
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