Co 102862 - CAS 181144-66-1
Catalog number: 181144-66-1
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C14H12FN3O2
Molecular Weight:
273.26
COA:
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Targets:
Sodium Channel
Description:
Co 102862, also known as V102862, an orally active anticonvulsant with robust activity, is a potent, broad-spectrum state-dependent inhibitor of mammalian voltage-gated Na+ channels with ~ 80-fold higher affinity for inactivated Na+ channels compared to channels in the resting state.
Purity:
>99 %
Appearance:
Pale yellow to white powder
Synonyms:
[[4-(4-fluorophenoxy)phenyl]methylideneamino]urea; 4-(4-fluorophenoxy)benzaldehyde semicarbazone; Co 102862; Co-102862; FPhOBal semicarbazone; 181144-66-1; 2-(4-(4-Fluorophenoxy)benzylidene)hydrazinecarboxamide; Hydrazinecarboxamide, 2-[[4-(4-fluorophenoxy)phenyl]methylene]-
Solubility:
Soluble to 100 mM in DMSO
MSDS:
Inquire
InChIKey:
MHUUDVZSPFRUSK-UHFFFAOYSA-N
InChI:
1S/C14H12FN3O2/c15-11-3-7-13(8-4-11)20-12-5-1-10(2-6-12)9-17-18-14(16)19/h1-9H,(H3,16,18,19)
Canonical SMILES:
C1=CC(=CC=C1C=NNC(=O)N)OC2=CC=C(C=C2)F
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Chemical Structure

CAS 181144-66-1 Co 102862

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