|Targets||mGluR | NMDA Receptor|
|Description||cis-ACPD has been found to be a potent NMDA receptor agonist as well as a mGluR agonist.|
|Purity||≥98% by HPLC|
Conantokin-T is a non-competitive NMDA receptor antagonist with IC50 value of 0.4 μM. It inhibits Ca2+ influx and glutamate-induced toxicity in central nervous ...
ZD 9379 is an antagonist of glycine site on the NMDA receptor, displaying neuroprotective effects. ZD 9379 reduces infarct size and frequency of spreading depre...
(RS)-MCPG Disodium Salt
(RS)-MCPG disodium salt is a non-selective group I/II metabotropic glutamate receptor antagonist.
MDL 105519, a ligand selective for the glycine binding site of NMDA receptor, was shown that completely inhibited the binding of [3H]glycine to rat brain membra...
Mephenesin is an NMDA receptor antagonist, is a centrally acting muscle relaxant.
(2R,4R)-APDC is a selective and relatively potent group II mGluR agonist (EC50 = 0.4, 0.4, > 100, > 100, > 300 and > 300 μM for human mGlu2, mGlu3, mGlu1, mGlu5...
BAY 36-7620 elective mGlu1 receptor non-competitive antagonist (IC50 = 0.16 μM) with inverse agonist activity.
Desmethyl-YM 298198 is a derivative of YM 298198, a selective antagonist of mGlu1.