|Description||cis-ACBD has been found to be a potent inhibitor of EAAT.|
|Purity||≥98% by HPLC|
cis-ACBD has been found to be a potent inhibitor of EAAT.
(±)-HIP-A is a potent and non-competitive excitatory amino acid transporter (EAAT) blocker. (±)-HIP-A displays no affinity for NMDA and metabotropic glutamate r...
TFB-TBOA is a glial glutamate transporter EAAT1 and EAAT2 inhibitor (IC50 = 17, 22 and 300 nM for EAAT2, EAAT1 and EAAT3, respectively). TFB-TBOA exhibits no ef...
L-TBOA is a potent and competitive blocker of human excitatory amino acid transporters (EAAT1-3; IC50 values 23 µM, 3.8 µM, 7.0 µM for EAAT1, EAAT2, and EAAT3, ...
LDN-212320 is a glutamate transporter EAAT2 activator. It increases expression of glutamate transporter EAAT2 in PA-EAAT2 cells and displays neuroprotective act...
WAY 213613 is a potent and non-substrate inhibitor of EAAT2 (GLT-1), displaying > 44-fold selectivity over EAAT1 and EAAT3 (IC50 = 85, 3787 and 5004 nM for EAAT...
DL-TBOA is a competitive and non-transportable inhibitor of excitatory amino acid transporters (IC50 = 70, 6, and 6 μM for EAAT1, EAAT2 and EAAT3, respectively)...
Dihydrokainic acid has been found to be an EAAT2(GLT1)-selective non-transportable inhibitor of L-glutamate and L-aspartate uptake.