Cilobradine hydrochloride - CAS 186097-54-1
Catalog number:
186097-54-1
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C28H39ClN2O5
Molecular Weight:
519.07
COA:
Inquire
Targets:
HCN Channel
Description:
Cilobradine hydrochloride, also called as DK-AH 269, a benzazepinone derivative, is an HCN Channel blocker that might be beneficial in the treatment of cardiovascular diseases, e.g. ischemia.
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Appearance:
White solid
Synonyms:
3-[[(3S)-1-[2-(3,4-dimethoxyphenyl)ethyl]piperidin-3-yl]methyl]-7,8-dimethoxy-2,5-dihydro-1H-3-benzazepin-4-one;hydrochloride 1,3,4,5-tetrahydro-7,8-dimethoxy-3-((1-(2-(3,4-dimethoxyphenyl)ethyl)-3-piperidinyl)methyl)-2H-3-benzazepin-2-one hydrochloride D
Solubility:
Soluble to 10 mM in H2O
Storage:
Store in a cool and dry place and at 0 - 4℃ for short term (days to weeks) or -74℃ for long term (months to years).
MSDS:
Inquire
Shelf Life:
2 years
InChIKey:
MTAKUIYCCYKGJJ-BOXHHOBZSA-N
InChI:
1S/C28H38N2O5.ClH/c1-32-24-8-7-20(14-25(24)33-2)9-12-29-11-5-6-21(18-29)19-30-13-10-22-15-26(34-3)27(35-4)16-23(22)17-28(30)31;/h7-8,14-16,21H,5-6,9-13,17-19H2,1-4H3;1H/t21-;/m0./s1
Canonical SMILES:
COC1=C(C=C(C=C1)CCN2CCCC(C2)CN3CCC4=CC(=C(C=C4CC3=O)OC)OC)OC.Cl
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Chemical Structure

CAS 186097-54-1 Cilobradine hydrochloride

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