CI-1018 - CAS 245329-99-1
Catalog number: 245329-99-1
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C24H20N4O2
Molecular Weight:
396.44
COA:
Inquire
Targets:
Phosphodiesterase (PDE)
Description:
CI-1018 is a selective type 4 phosphodiesterase inhibitor associated with vasculitis. CI-1018 has been in development to suppress inflammation.
Purity:
>98%
Appearance:
Solid powder
Synonyms:
4-Pyridinecarboxamide, N-(3,4,6,7-tetrahydro-9-methyl-4-oxo-1-phenylpyrrolo(3,2,1-jk)(1,4)benzodiazepin-3-yl)-; CI-1018; CI-1018; CI-1018; UNII-05127JZ9KQ
MSDS:
Inquire
InChIKey:
KYFWUBJMTHVBIF-QFIPXVFZSA-N
InChI:
1S/C24H20N4O2/c1-15-13-18-9-12-28-21(18)19(14-15)20(16-5-3-2-4-6-16)26-22(24(28)30)27-23(29)17-7-10-25-11-8-17/h2-8,10-11,13-14,22H,9,12H2,1H3,(H,27,29)/t22-/m0/s1
Canonical SMILES:
CC1=CC2=C3C(=C1)C(=NC(C(=O)N3CC2)NC(=O)C4=CC=NC=C4)C5=CC=CC=C5
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