Chlorotrianisene - CAS 569-57-3
Catalog number:
569-57-3
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C23H21ClO3
Molecular Weight:
380.87
COA:
Inquire
Targets:
Estrogen Receptor/ERR
Description:
Chlorotrianisene is a powerful synthetic, non-steroidal estrogenic compound which is metabolized by liver microsomal enzymes primarily to the mono-O-demethylated derivative. It binds to the estrogen receptor on various estrogen receptor bearing cells. It was used for the treatment of menopause, deficiencies in ovary function, and prostate cancer. It belongs triphenylethylene group. It was derived from estrobin (DBE) and is a relatively weak estrogen. It is a selective estrogen receptor modulator (SERM), with predominantly estrogenic but also antiestrogenic effects, and was arguably the first SERM to ever be introduced. It has been listed.
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Purity:
95%
Appearance:
White powder
Synonyms:
1,1',1''-(1-Chloro-1-ethenyl-2-ylidene)-tris(4-methoxybenzene);1-[2-Chloro-1,2-bis(4-methoxyphenyl)vinyl]-4-methoxybenzene;Chlortrianisestrol;Chlortrianizen;Khlortrianizen;Hormonisene;Anisene;Metace;Rianil;Tace;1-[1-Chloro-2,2-bis(4-methoxyphenyl)ethenyl]
Solubility:
Soluble in DMSO, not in water
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
Chlorotrianisene was used for the treatment of menopause, deficiencies in ovary function, and prostate cancer.
Quality Standard:
In-house standard
Quantity:
Grams to Kilograms
Boiling Point:
514.2±45.0 °C | Condition: Press: 760 Torr
Melting Point:
114-116 °
Density:
1.168±0.06 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr
InChIKey:
BFPSDSIWYFKGBC-UHFFFAOYSA-N
InChI:
InChI=1S/C23H21ClO3/c1-25-19-10-4-16(5-11-19)22(17-6-12-20(26-2)13-7-17)23(24)18-8-14-21(27-3)15-9-18/h4-15H,1-3H3
Canonical SMILES:
COC1=CC=C(C=C1)C(=C(C2=CC=C(C=C2)OC)Cl)C3=CC=C(C=C3)OC
Current Developer:
Chlorotrianisene has been listed.
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CAS 569-57-3 Chlorotrianisene

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