CHF-4227 - CAS 444643-64-5
Catalog number:
444643-64-5
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C30H33NO4
Molecular Weight:
471.59
COA:
Inquire
Targets:
Estrogen Receptor/ERR
Description:
CHF-4227 is a selective estrogen receptor modulator, binds with high affinity to the human estrogen receptor-alpha and -beta (dissociation constant K(i) = 0.017 and 0.099 nM, respectively).
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Purity:
≥98%
Appearance:
Solid powder
Synonyms:
3-(4-methoxyphenyl)-4-(4-(2-(piperidin-1-yl)ethoxy)benzyl)-2H-chromen-7-ol;
Solubility:
Soluble in DMSO
Storage:
Store at -20 °C
MSDS:
Inquire
Application:
estrogen receptor modulator
Quality Standard:
Enterprise standard
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly.
Quantity:
Milligrams-Grams
InChIKey:
ZUDXUNPSRMREOJ-UHFFFAOYSA-N
InChI:
1S/C30H33NO4/c1-33-25-12-7-23(8-13-25)29-21-35-30-20-24(32)9-14-27(30)28(29)19-22-5-10-26(11-6-22)34-18-17-31-15-3-2-4-16-31/h5-14,20,32H,2-4,15-19,21H2,1H3
Canonical SMILES:
COc1ccc(cc1)C2=C(c3ccc(cc3OC2)O)Cc4ccc(cc4)OCCN5CCCCC5
Current Developer:
Chiesi Farmaceutici
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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