CGP 3466B maleate - CAS 200189-97-5
Catalog number: 200189-97-5
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C23H21NO5
Molecular Weight:
391.42
COA:
Inquire
Targets:
Others
Description:
CGP 3466B maleate, a potent anti-apoptotic drug, is an orally active glyceraldehyde-3-phosphate dehydrogenase (GAPDH) inhibitor. CGP 3466B maleate was tested in clinical trials for its ability to help treat Parkinson's disease (PD) and amyotrophic lateral sclerosis (ALS) but the clinical trials have been terminated due to lack of benefit.
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Purity:
>99 %
Appearance:
Solid powder
Synonyms:
N-(benzo[b][1]benzoxepin-5-ylmethyl)-N-methylprop-2-yn-1-amine;but-2-enedioic acid; Omigapil maleate; CGP 3466B; CGP-3466B; CGP3466B; TCH-346; TCH 346; TCH346; Omigapil maleate
MSDS:
Inquire
InChIKey:
SQAZQLMBEHYFJA-UHFFFAOYSA-N
InChI:
1S/C19H17NO.C4H4O4/c1-3-12-20(2)14-16-13-15-8-4-6-10-18(15)21-19-11-7-5-9-17(16)19;5-3(6)1-2-4(7)8/h1,4-11,13H,12,14H2,2H3;1-2H,(H,5,6)(H,7,8)
Canonical SMILES:
CN(CC#C)CC1=CC2=CC=CC=C2OC3=CC=CC=C31.C(=CC(=O)O)C(=O)O
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CAS 200189-97-5 CGP 3466B maleate

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