CFI-400936 - CAS 1338793-07-9
Catalog number: 1338793-07-9
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C25H27N5O3S
Molecular Weight:
477.58
COA:
Inquire
Targets:
Others
Description:
CFI-400936 is a selective proteine kinase TTK inhibitor with IC50 value of 3.6nM. It demonstrates good activity in cell based assay and selectivity against a panel of human kinases. CFI-400936 shows potential anticancer activity.
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Purity:
98%
Appearance:
Powder
Synonyms:
2-(dimethylamino)-2-(2-ethylphenyl)-N-(3-(3-sulfamoylphenyl)-1H-indazol-5-yl)acetamide
Solubility:
Soluble in DMSO
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
anticancer
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
Canonical SMILES:
O=C(NC1=CC2=C(NN=C2C3=CC=CC(S(=O)(N)=O)=C3)C=C1)C(N(C)C)C4=CC=CC=C4CC
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