|Description||Ceftaroline fosamil, a cephalosporin antibiotic, is active against methicillin-resistant Staphylococcus aureus (MRSA) and Gram-positive bacteria.|
|Synonyms||(6R,7R)-7-[[(2Z)-2-ethoxyimino-2-[5-(phosphonoamino)-1,2,4-thiadiazol-3-yl]acetyl]amino]-3-[[4-(1-methylpyridin-1-ium-4-yl)-1,3-thiazol-2-yl]sulfanyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate; TAK 599; TAK599; TAK-599; PPI 0903; PP 0903; PPI-0903; T-91825; T 91825; T91825; Ceftaroline fosamil; Teflaro; Zinforo|
Novobiocin Sodium is a very potent bacterial DNA gyrase and human organic anion transporters with Ki of 14.87 ± 0.40 μM for hOAT1, 4.77 ± 1.12 μM for hOAT3 and ...
Enrofloxacin is a fluoroquinolone antibiotic acting by inhibiting bacterial DNA gyrase (a type-II topoisomerase), thereby preventing DNA supercoiling and DNA sy...
Cefpodoxime Proxetil is a third generation cephalosporin, ester prodrug of the active free acid metabolite Cefpodoxime. Cefpodoxime is active against most Gram-...
Garenoxacin Mesylate hydrate
Garenoxacin Mesylate hydrate is the Mesylate hydrate salt form of Garenoxacin. Garenoxacin, also called as BMS 284756, a new desfluoro(6)quinolone, is a topoiso...
Ampicillin is a beta-lactam antibiotic that is part of the aminopenicillin family and is roughly equivalent to its successor, amoxicillin in terms of spectrum a...
Biapenem (INN) is a carbapenem antibiotic. It has in vitro activity against anaerobes.
Ribocil, a newly developed riboswitches chemical modulator, could selectively restrain the expression of GFP and probably influence bacterial cell growth. IC50:...
Sulfisomidin, closely related to sulfadimidine, is a sulfonamide antibacterial.
Olsalazine Sodium is an anti-inflammatory prodrug, which consists of two 5-ASA moieties linked by an azo bond. It is used in the treatment of inflammatory bowel...
The diisethionate salt form of Pentamidine, an amidine derivative, has been found to have antiprotozoal and antifungal effect and could be commonly used against...
Nitroxoline is a urinary antibacterial agent had proven to be very effective at combating biofilm infections.
Sarafloxacin is a quinolone antibiotic drug, inhibiting the topoisomerase II ligase domain.
KKL-10 is a small-molecule ribosome rescue inhibitor with exceptional antimicrobial activity against both attenuated and fully virulent strains of F. tularensis...
Fleroxacin is a bactericidal drug that inhibits bacterial DNA gyrase and topoisomerase IV. Like other quinolones and fluoroquinolones, it eradicates bacteria by...
Thiamphenicol is an antimicrobial antibiotic and a methyl-sulfonyl analogue of chloramphenicol.
Ceftiofur sodium, one of the third generation antibiotics, is a cephalosporin based antibacterial compound that has been approved to be used in veterinary medic...
NITD-304, an indole derivative, has been found to be an antitubercular agent that could be effective through influencing multidrug-resistant mycobacterium tuber...
Dextrorotation nimorazole phosphate este
The organic phosphate form of Dextrorotary morpholine ornidazole, an effective anti-parasitic agent, has been found to have better tolerance as one of the fourt...
Ofloxacin is a synthetic broad-spectrum antimicrobial agent.
Tebipenem(LJC-11036) is a broad spectrum orally administered antibiotic; exhibits slow tight-binding inhibition at low micromolar concentrations versus the chro...