CCG215022 - CAS 1813527-81-9
Category: Inhibitor
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Molecular Formula:
Molecular Weight:
CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor (IC50s= 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, GRK5 and GRK1, respectively), with good selectivity against other closely related kinases such as GRK1 and PKA.
Solid powder
4-(4-fluoro-3-((pyridin-2-ylmethyl)carbamoyl)phenyl)-N-(1H-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide; CCG215022; CCG 215022; CCG-215022.
Store in a cool and dry place (or refer to the Certificate of Analysis).
Boiling Point:
783.2±60.0 °C at 760 Torr
1.422±0.06 g/cm3
Canonical SMILES:
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CAS 1813527-81-9 CCG215022

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