|Description||CBL0137 is a metabolically stable curaxin that activates p53 with an EC50 value of 0.37 µM and inhibits NF-κB with an EC50 of 0.47 µM. It also inhibits histone chaperone FACT (facilitates chromatin transcription) and MYC signal.|
|B0084-284751||2.5 mg||$198||In stock|
|Synonyms||CBL-0137; Curaxin 137; 1,1'-(9-(2-(Isopropylamino)ethyl)-9H-carbazole-3,6-diyl)diethanone; 1-[6-acetyl-9-[2-(propan-2-ylamino)ethyl]carbazol-3-yl]ethanone|
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