CBB1003 - CAS 1379573-88-2
Catalog number:
1379573-88-2
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C25H31N9O4
Molecular Weight:
521.57
COA:
Inquire
Targets:
Histone Demethylase
Description:
CBB1003, a piperazine derivative, has been found to be a histone demethylase LSD1 inhibitor that could restrain the proliferation and colony formation of CRC cell in mice. IC50: 10.54 uM.
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Purity:
98%
Appearance:
Powder
Synonyms:
CBB1003; SCHEMBL16273292; CS-3476
Solubility:
10 mM in DMSO
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
CBB1003 has been found to be a histone demethylase LSD1 inhibitor that could restrain the proliferation and colony formation of CRC cell in mice.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
SKTVJNLOILHEKO-UHFFFAOYSA-N
InChI:
InChI=1S/C25H31N9O4/c26-22(27)18-1-3-19(4-2-18)23(35)31-9-11-32(12-10-31)24(36)20-13-17(14-21(15-20)34(37)38)16-30-5-7-33(8-6-30)25(28)29/h1-4,13-15H,5-12,16H2,(H3,26,27)(H3,28,29)
Canonical SMILES:
C1CN(CCN1CC2=CC(=CC(=C2)C(=O)N3CCN(CC3)C(=O)C4=CC=C(C=C4)C(=N)N)[N+](=O)[O-])C(=N)N
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