|Description||Santacruzamate A (CAY10683) is a potent and selective HDAC inhibitor with IC50 of 119 pM for HDAC2, >3600-fold selectivity over other HDACs.|
Brefeldin A is a fungal metabolite and blocks the forward transport between the endoplasmic reticulum and Golgi apparatus, Brefeldin A causes an impaired distri...
NSC 663284 is a potent, irreversible, cell permeable and mixed competitive Cdc25 dual specificity phosphatases inhibitor (IC50= 0.21 μM), and poorly inhibits ot...
OTX008, a calixarene derivative, is a galectin-1 (Gal-1) inhibitor with potential anti-angiogenic and antineoplastic activities. In vitro, OTX008 effects in a p...
6-O-α-D-Maltosyl-β-cyclodextrin is a cellular cholesterol modifier which can form soluble inclusion complex with cholesterol and is much less cytotoxic to human...
10-Undecylenic Acid, a long-chain fatty acid substance, could be used as a monomer in the polymerization and also a raw material in the syntheses of Pheromone (...
CP-467688 is a microsomal triglyceride transfer protein inhibitor used in atherosclerosis therapy.
Eicosapentaenoic acid (EPA) is an omega-3 fatty acid.
Nabumetone is a non-steroidal anti-inflammatory drug and its active metabolite inhibits the COX.
Maprotiline HCl is a selective noradrenalin re-uptake inhibitor and a tetracyclic antidepressant.
FR 121196 is a potential antidementia drug originated by Fujisawa. Mechanism of Action is not undefined. FR 121196 can ameliorate the impaired memory of rat in ...
Tinyatoxin is a neurotoxin, acting via vanilloid receptors of sensory nerves.
Minocycline is a broad-spectrum tetracycline antibiotic, which has a broader spectrum than the other members of the group. It has a 7-dimethylamino and lacking ...
Peiminine and DXS significantly reduced alveolar inflammation and pulmonary interstitial inflammation in rats with bleomycin-induced lung injury. peiminine inhi...
Used as a substrate for the detection of sialidase-like enzyme in screening of enzymes, studying physiological activities of gangliosides, and recombinant techn...
Mycophenolate mofetil hydrochloride
Mycophenolate mofetil is a non-competitive, selective and reversible inhibitor of inosine monophosphate dehydrogenase I/II with IC50 of 39 nM and 27 nM, respect...
D-Xylose, a natural product, is used in diagnostic malabsorption tests as well as in the production of Furfural.
Bucetin, a phenacetin analog, has antipyretic and analgesic effect. It has been discontinued for showing renal toxicity.
Ocaphane is a strong antitumor agent used on a number of animal tumors along with fairly toxic to hemopoietic organs.
BMS711939 is a selective and potent peroxisome proliferator-activated receptor α(PPARα) agonist with EC50 value of 4 nM for human PPARα. It is >1000-fold select...
Eflornithine hydrochloride is a drug found to be effective in the treatment of facial hirsutism. It is a "suicide inhibitor," irreversibly binding to Ornithine ...