CaMKII-IN-1 - CAS 1208123-85-6
Catalog number: 1208123-85-6
Category: Inhibitor
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Molecular Formula:
C29H30ClN5O2S
Molecular Weight:
548.1
COA:
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Targets:
CaMK-II
Description:
CaMKII-IN-1 is a potent and highly selective CaMKII inhibitor with IC50 of 63 nM; significantly high selectivity against CaMKIV, MLCK, p38a, Akt1, and PKC.
Purity:
>98%
Synonyms:
CaMKII-IN-1
MSDS:
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InChIKey:
LGUUETDTMQTHML-UHFFFAOYSA-N
InChI:
InChI=1S/C29H30ClN5O2S/c1-21-25(30)13-8-14-27(21)38(36,37)34-28-24-20-35(19-23-11-6-3-7-12-23)18-16-26(24)32-29(33-28)31-17-15-22-9-4-2-5-10-22/h2-14H,15-20H2,1H3,(H2,31,32,33,34)
Canonical SMILES:
CC1=C(C=CC=C1Cl)S(=O)(=O)NC2=NC(=NC3=C2CN(CC3)CC4=CC=CC=C4)NCCC5=CC=CC=C5
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Chemical Structure

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