BYK 49187 - CAS 163120-31-8
Category: Inhibitor
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Molecular Formula:
C19H21N5O
Molecular Weight:
335.4
COA:
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Targets:
PARP
Description:
BYK 49187 is a non-selective PARP inhibitor (pIC50 = 8.36 and 7.50 for cell-free recombinant PARP-1 and murine PARP-2, respectively).
Brife Description:
PARP inhibitor
Purity:
≥98% by HPLC
Synonyms:
BYK 49187; BYK49187; BYK-49187; 4,5-Dihydro-2-[4-(4-methyl-1H-imidazol-4-yl)-1-piperidinyl]-6H-imidazo[4,5,1-ij]quinolin-6-one
MSDS:
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InChIKey:
YKJJROIKVYSPDH-UHFFFAOYSA-N
InChI:
InChI=1S/C19H21N5O/c1-12-17(21-11-20-12)13-5-8-23(9-6-13)19-22-15-4-2-3-14-16(25)7-10-24(19)18(14)15/h2-4,11,13H,5-10H2,1H3,(H,20,21)
Canonical SMILES:
CC1=C(N=CN1)C2CCN(CC2)C3=NC4=CC=CC5=C4N3CCC5=O
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Chemical Structure

CAS 163120-31-8 BYK 49187

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