|Description||BYK 204165 is a potent and selective poly(ADP-ribose) polymerase (PARP)-1 inhibitor (pIC50 = 5.38 and 7.35 for PARP-2 and PARP-1, respectively). BYK 204165 is 100-fold more potent for PARP-1 than PARP-2.|
|Brife Description||PARP-1 inhibitor|
|Purity||≥99% by HPLC|
|Synonyms||PARP Inhibitor XIV; RT 017290; 4-[(1-Methyl-1H-pyrrol-2-yl)methylene]-1,3(2H,4H)-isoquinolinedione|
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