BYK 204165 - CAS 1104546-89-5
Category: Inhibitor
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Molecular Formula:
C15H12N2O2
Molecular Weight:
252.27
COA:
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Targets:
PARP
Description:
BYK 204165 is a potent and selective poly(ADP-ribose) polymerase (PARP)-1 inhibitor (pIC50 = 5.38 and 7.35 for PARP-2 and PARP-1, respectively). BYK 204165 is 100-fold more potent for PARP-1 than PARP-2.
Brife Description:
PARP-1 inhibitor
Purity:
≥99% by HPLC
Synonyms:
PARP Inhibitor XIV; BYK204165; BYK-204165; BYK 204165; RT-017290; RT017290; RT 017290. 4-[(1-Methyl-1H-pyrrol-2-yl)methylene]-1,3(2H,4H)-isoquinolinedione
MSDS:
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InChIKey:
BTYSIDSTHDDAJW-LCYFTJDESA-N
InChI:
InChI=1S/C15H12N2O2/c1-17-8-4-5-10(17)9-13-11-6-2-3-7-12(11)14(18)16-15(13)19/h2-9H,1H3,(H,16,18,19)/b13-9-
Canonical SMILES:
CN1C=CC=C1C=C2C3=CC=CC=C3C(=O)NC2=O
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Chemical Structure

CAS 1104546-89-5 BYK 204165

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