Bromosporine - CAS 1619994-69-2
Catalog number: 1619994-69-2
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C17H20N6O4S
Molecular Weight:
404.44
COA:
Inquire
Targets:
BET Bromodomain
Description:
Bromosporine, a broad spectrum inhibitor for bromodomains which play a key role in many cellular processes, is a chemical probe for bromodomain functional assays so that it is very helpful in elucidating further biological roles of reader domains. IC50: B
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Appearance:
Solid powder
Synonyms:
ethyl N-[6-[3-(methanesulfonamido)-4-methylphenyl]-3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-8-yl]carbamate Bromosporine 1619994-69-2 ethyl (3-methyl-6-(4-methyl-3-(methylsulfonamido)phenyl)-[1,2,4]triazolo[4,3-b]pyridazin-8-yl)carbamate Bromorsporine GTPL
Solubility:
DMSO: ≥ 51.7 mg/mL
Storage:
Store in a cool and dry place and at 0 - 4℃ for short term (days to weeks) or -32℃ for long term (months to years).
MSDS:
Inquire
Shelf Life:
2 years
Quantity:
Grams-Kilos
Density:
1.46±0.1 g/cm3
InChIKey:
UYBRROMMFMPJAN-UHFFFAOYSA-N
InChI:
1S/C17H20N6O4S/c1-5-27-17(24)18-15-9-14(21-23-11(3)19-20-16(15)23)12-7-6-10(2)13(8-12)22-28(4,25)26/h6-9,22H,5H2,1-4H3,(H,18,24)
Canonical SMILES:
CCOC(=O)NC1=CC(=NN2C1=NN=C2C)C3=CC(=C(C=C3)C)NS(=O)(=O)C
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Chemical Structure

CAS 1619994-69-2 Bromosporine

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