BRN-103 - CAS 1346265-80-2
Catalog number:
1346265-80-2
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C24H25ClN4O
Molecular Weight:
420.93
COA:
Inquire
Targets:
VEGFR
Description:
BRN-103 can suppress the phosphorylation of vascular endothelial growth factor (VEGF) receptor 2. It can also inhibit the activations of AKT and eNOS. These results show that BRN-103 inhibits VEGF-mediated angiogenesis signaling in human endothelial cells.
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Purity:
98%
Appearance:
Powder
Synonyms:
2-((1-benzylpiperidin-4-yl)amino)-N-(3-chlorophenyl)nicotinamide
Solubility:
Soluble in DMSO
Storage:
-20°C Freezer
MSDS:
Inquire
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Gram
InChI:
InChI=1S/C24H25ClN4O/c25-19-8-4-9-21(16-19)28-24(30)22-10-5-13-26-23(22)27-20-11-14-29(15-12-20)17-18-6-2-1-3-7-18/h1-10,13,16,20H,11-12,14-15,17H2,(H,26,27)(H,28,30)
Canonical SMILES:
O=C(C1=CC=CN=C1NC2CCN(CC3=CC=CC=C3)CC2)NC4=CC=CC(Cl)=C4
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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