BRL 50481 - CAS 433695-36-4
Catalog number: 433695-36-4
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C9H12N2O4S
Molecular Weight:
244.27
COA:
Inquire
Targets:
Phosphodiesterase (PDE)
Description:
BRL 50481 is a potent, selective substrate-competitive inhibitor of phosphodiesterase (PDE) 7 (Ki = 180 nM).
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Purity:
≥95%
Appearance:
Off-White Solid
Synonyms:
3-(N,N-Dimethylsulfonamido)-4-methylnitrobenzene, 5-Nitro-2-N,N-trimethylbenzenesulfonamide;
Solubility:
Soluble in DMSO
Storage:
Store at -20 °C
MSDS:
Inquire
Application:
A PDE7 inhibitor that has acceptable selectivity for in vivo studies.
Quality Standard:
Enterprise standard
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly.
Quantity:
Milligrams-Grams
Melting Point:
72-74 °C
InChIKey:
IFIUFCJFLGCQPH-UHFFFAOYSA-N
InChI:
1S/C9H12N2O4S/c1-7-4-5-8(11(12)13)6-9(7)16(14,15)10(2)3/h4-6H,1-3H3
Canonical SMILES:
CC1=C(S(N(C)C)(=O)=O)C=C([N+]([O-])=O)C=C1
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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