|Description||Bretazenil is a partial agonist at the GABAA benzodiazepine site (EC50 = 10 nM at α1β1γ2 receptors) that potentiates GABA responses on α4β3γ2 cells. Bretazenil is potentially used for the treatment of anxiety disorders.|
|Brife Description||GABAA receptor agonist|
|Purity||≥98% by HPLC|
|Synonyms||(13aS)-8-Bromo-11,12,13,13a-tetrahydro-9-oxo-9H-imidazo[1,5-a]pyrrolo[2,1-c][1,4]benzodiazepine-1-carboxylic acid 1,1-dimethylethyl ester; Ro 16-6028; Ro 16 6028; Ro16-6028; Ro 166028; Ro 166028; Ro166028; Ro 16-6028/000; Bretazenil|
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