|Targets||5-HT Receptor | Sigma Receptor|
|Description||BMY 14802 hydrochloride is a potent sigma receptor antagonist (IC50 = 112 nM) with weak affinity for 5-HT1A and α1 receptors. BMY 14802 is potentially used as an atypical antipsychotic agent for schizophrenia treatment.|
|Brife Description||sigma receptor antagonist|
|Purity||≥98% by HPLC|
|Related CAS||105565-56-8 (free base)|
|Synonyms||BMS-181100 hydrochloride; BMY 14802 HCl; α-(4-Fluorophenyl)-4-(5-fluoro-2-pyrimidinyl)-1-piperazinebutanol hydrochloride|
|Application||potential atypical antipsychotic agent|
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BMY 14802 hydrochloride
BMY 14802 hydrochloride is a potent sigma receptor antagonist (IC50 = 112 nM) with weak affinity for 5-HT1A and α1 receptors. BMY 14802 is potentially used as a...
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