BMS585248 - CAS 619331-12-3
Catalog number: 619331-12-3
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C22H18FN7O3
Molecular Weight:
447.43
COA:
Inquire
Targets:
HIV
Description:
BMS585248 is a highly potent and novel human immunodeficiency virus type 1 (HIV-1) attachment inhibitor with 4-fluoro-6-azaindole core heterocycles. It targets the viral envelope protein gp120. It showed much improved in vitro potency and pharmacokinetic properties than the previous clinical candidate BMS488043.
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Purity:
98%
Appearance:
Solid powder
Synonyms:
BMS-585248;1,2-Ethanedione, 1-(4-benzoyl-1-piperazinyl)-2-(4-fluoro-7-(1H-1,2,3-triazol-1-yl)-1H-pyrrolo(2,3-c)pyridin-3-yl)-;1-(4-Benzoylpiperazin-1-yl)-2-[4-fluoro-7-(triazol-1-yl)-1H-pyrrolo[2,3-c]pyridin-3-yl]ethane-1,2-dione
Solubility:
Soluble in DMSO, not in water
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
BMS585248 targets the viral envelope protein gp120.
Quality Standard:
In-house standard
Quantity:
Milligrams-Grams
Boiling Point:
733.0±70.0 °C | Condition: Press: 760 Torr
Density:
1.54±0.1 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr
InChIKey:
YILIMUKOYIOIAY-UHFFFAOYSA-N
InChI:
InChI=1S/C22H18FN7O3/c23-16-13-25-20(30-7-6-26-27-30)18-17(16)15(12-24-18)19(31)22(33)29-10-8-28(9-11-29)21(32)14-4-2-1-3-5-14/h1-7,12-13,24H,8-11H2
Canonical SMILES:
C1CN(CCN1C(=O)C2=CC=CC=C2)C(=O)C(=O)C3=CNC4=C3C(=CN=C4N5C=CN=N5)F
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