BMS-779788 - CAS 918348-67-1
Catalog number: B0084-284850
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C28H29ClN2O3S
Molecular Weight:
509.061
COA:
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Targets:
LXR
Description:
BMS-779788 is a LXR partial agonist with IC50 values of 68 nM and 14 nM for LXRα and LXRβ respectively. BMS-779788 induces LXR target genes in blood in vivo with EC50 value of 610 nM, and significantly increases plasma triglyceride and LDL cholesterol.
Ordering Information
Catalog Number Size Price Stock Quantity
B0084-284850 25 mg $198 In stock
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Brife Description:
LXR partial agonist
Synonyms:
XL-652; 2-[2-[2-(2-chlorophenyl)propan-2-yl]-1-[4-(3-methylsulfonylphenyl)phenyl]imidazol-4-yl]propan-2-ol
MSDS:
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InChIKey:
JLPURTXCSILYLW-UHFFFAOYSA-N
InChI:
InChI=1S/C28H29ClN2O3S/c1-27(2,23-11-6-7-12-24(23)29)26-30-25(28(3,4)32)18-31(26)21-15-13-19(14-16-21)20-9-8-10-22(17-20)35(5,33)34/h6-18,32H,1-5H3
Canonical SMILES:
CC(C)(C1=CC=CC=C1Cl)C2=NC(=CN2C3=CC=C(C=C3)C4=CC(=CC=C4)S(=O)(=O)C)C(C)(C)O
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