BMS-505130 - CAS 859230-84-5
Catalog number:
859230-84-5
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C19H21N3O4
Molecular Weight:
355.39
COA:
Inquire
Targets:
Others
Description:
BMS-505130 is a selective serotonin transport inhibitor with Ki of 0.18 nM. Ki value for binding to the norepinephrine is 4.6 mM and for dopamine transporters is 2.1 mM.
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Purity:
98%
Appearance:
Powder
Synonyms:
UNII-E892TW82D9; E892TW82D9;1H-Indole-5-carbonitrile, 3-((1S,2S)-2-((dimethylamino)methyl)cyclopropyl)-, (2Z)-2-butenedioate (1:1)
Solubility:
Soluble in DMSO
Storage:
-20℃ Freezer
MSDS:
Inquire
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
QYXJWBDKQAIHJM-ZMPXXIOZSA-N
InChI:
1S/C15H17N3.C4H4O4/c1-18(2)9-11-6-12(11)14-8-17-15-4-3-10(7-16)5-13(14)15;5-3(6)1-2-4(7)8/h3-5,8,11-12,17H,6,9H2,1-2H3;1-2H,(H,5,6)(H,7,8)/b;2-1-/t11-,12+;/m1./s1
Canonical SMILES:
CN(C)C[C@H]1C[C@@H]1c2c[nH]c3c2cc(cc3)C#N.C(=C\C(=O)O)\C(=O)O
Current Developer:
Originator Bristol-Myers Squibb
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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