BMS-354326 - CAS 708258-16-6
Catalog number: 708258-16-6
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C28H40N4O5
Molecular Weight:
512.65
COA:
Inquire
Targets:
Ser/Thr Protease
Description:
BMS-354326 is a tryptase inhibitor with IC50 value of 1.8 nM. It has excellent selectivity against trypsin and most other related serine proteases.
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Purity:
98%
Appearance:
Powder
Synonyms:
CHEMBL306448; BDBM50144532;(2S,3R)-4-oxo-1-((4-(1-oxo-6-phenylhexyl)-1-piperazinyl)carbonyl)-3-(2-(3-piperidinyl)ethyl)- 2-Azetidinecarboxylic acid,
Solubility:
Soluble in DMSO
Storage:
-20℃ Freezer
MSDS:
Inquire
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
XVYFBYVSZOCXRJ-OMQKAAQBSA-N
InChI:
1S/C28H40N4O5/c33-24(12-6-2-5-10-21-8-3-1-4-9-21)30-16-18-31(19-17-30)28(37)32-25(27(35)36)23(26(32)34)14-13-22-11-7-15-29-20-22/h1,3-4,8-9,22-23,25,29H,2,5-7,10-20H2,(H,35,36)/t22?,23-,25+/m1/s1
Canonical SMILES:
c1ccc(cc1)CCCCCC(=O)N2CCN(CC2)C(=O)N3[C@@H]([C@H](C3=O)CCC4CCCNC4)C(=O)O
Current Developer:
Bristol-Myers Squibb
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