|Targets||Checkpoint Kinase (Chk)|
|Description||BML-277 is a selective APT-competitive inhibitor of the DNA damage response signaling enzyme CHK2 ( IC50 =15 nM).|
|Synonyms||Chk2 Inhibitor II; 2-[4-(4-chlorophenoxy)phenyl]-3H-benzimidazole-5-carboxamide;|
|Solubility||Soluble in DMSO|
|Storage||Store at -20 °C|
|Application||A selective APT-competitive inhibitor|
|Quality Standard||Enterprise Standard|
|Shelf Life||As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly|
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